V2EX bioavailability

Bioavailability

释义 Definition

生物利用度:指药物或其他物质进入体内后,以未被改变的形式到达全身血液循环的比例与速度。口服药通常会因吸收不完全或“首过效应”(肝脏代谢)而降低生物利用度。(该词在营养学中也可指营养素被吸收利用的程度。)

发音 Pronunciation

/ba.o.ve.lbl..ti/
/ba..ve.lbl..ti/

例句 Examples

The tablet has low bioavailability when taken with food.
这片药与食物同服时生物利用度较低。

Because of extensive first-pass metabolism, the drug’s oral bioavailability is much lower than its intravenous bioavailability.
由于明显的首过代谢,这种药物的口服生物利用度远低于静脉给药的生物利用度。

词源 Etymology

由 **bio-**(生命、与生物相关)+ availability(可获得性、可用性)构成。原意可理解为“在生物体内可被利用的程度”,后来在药理学与药代动力学中固定指向“进入体循环的比例与速度”。

相关词 Related Words

文献与著作 Literary Works

  • Goodman & Gilman’s The Pharmacological Basis of Therapeutics
  • Katzung & Trevor’s Basic & Clinical Pharmacology
  • Rang & Dale’s Pharmacology
  • Rowland and Tozer’s Clinical Pharmacokinetics and Pharmacodynamics
  • U.S. FDA 指南:Bioavailability and Bioequivalence Studies Submitted in NDAs or INDs General Considerations
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