V2EX allosteric regulation

Allosteric Regulation

释义 Definition

变构调节:指酶或受体蛋白在非活性位点(变构位点)与某种分子(变构效应物)结合后,引起蛋白构象变化,从而增强或抑制其活性的一种调控方式。常见于代谢途径的反馈调控。
(该术语也常扩展用于描述蛋白质功能被远端位点结合事件所调控的现象。)

发音 Pronunciation (IPA)

/lstrk rjlen/

例句 Examples

Allosteric regulation helps enzymes respond quickly to changes in the cell.
变构调节帮助酶快速响应细胞内环境的变化。

In many metabolic pathways, allosteric regulation enables feedback inhibition, where the final product binds to an enzyme and slows the pathway down.
在许多代谢通路中,变构调节使反馈抑制成为可能:终产物与某种酶结合,从而减慢整个通路的反应速度。

词源 Etymology

allosteric 来自希腊语:*allo-*(“其他的、不同的”)+ stereos(“立体的、空间结构的”),强调“在不同位置发生结合并改变空间构象”。regulation 源自拉丁语 regulare(“引、规范、调节”)。合起来表示“通过不同位点的结合来调节活性”。

相关词 Related Words

文学与经典著作 Literary Works

  • Monod, Wyman & Changeux (1965), “On the nature of allosteric transitions: a plausible model”(提出经典的 MWC 变构模型,讨论变构调节的理论基础)
  • Berg, Tymoczko & Stryer, Biochemistry(《生物化学》,多版教材均系统讲解变构调节与代谢控制)
  • Lehninger, Principles of Biochemistry(《莱宁格生物化学原理》,常以实例说明酶的变构调节与反馈抑制)
  • Alberts et al., Molecular Biology of the Cell(《细胞的分子生物学》,在细胞调控与信号通路语境中涉及变构调节)
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