V2EX allosteric

Allosteric

释义 Definition

变构的;(指酶/蛋白质)别构调节的。
常用于生物化学与分子生物学中,描述一种现象:分子在非活性位点(别构位点)结合后,引起蛋白质构象改变,从而增强或抑制其功能(例如酶活性或受体信号)。

发音 Pronunciation (IPA)

/lstrk/

例句 Examples

Allosteric inhibitors can slow an enzyme down.
变构抑制剂可以减慢酶的反应速度。

By binding to an allosteric site, the drug changes the receptor’s shape and reduces its signaling without blocking the main binding site.
这种药物与别构位点结合后,会改变受体的形状,在不直接阻塞主要结合位点的情况下减弱信号传递。

词源 Etymology

allosteric 来自希腊语构词:allo-(“其他的、不同的”)+ stereos(“立体的、空间结构”)。字面含义接近“另一种空间构型/结构”,用于强调:分子结合发生在“另一个位置”,却能通过结构变化影响功能。该术语在20世纪中期随着酶的调控理论发展而广泛使用。

相关词 Related Words

文献与作品 Literary / Notable Works

  • Lehninger Principles of Biochemistry(《雷宁格生物化学原理》)
  • Molecular Biology of the Cell(《细胞的分子生物学》)
  • Biochemistry by Berg, Tymoczko & Stryer(《斯崔尔生物化学》)
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