V2EX pde3

PDE3

Definition / 释义

PDE3phosphodiesterase 3(磷酸二酯酶3) 的缩写,指一类分解细胞内信号分子(主要是 cAMP,也可影响 cGMP)的酶。它在心肌收缩、血管舒张、血小板功能等生理过程中很重要;相关的 PDE3 抑制剂可用于某些心血管或血小板相关疾病的治疗。

Pronunciation / 发音

/pidii θri/

Examples / 例句

PDE3 helps regulate cAMP levels in cells.
PDE3 有助于调节细胞内的 cAMP 水平。

In cardiology, PDE3 inhibitors can increase cardiac contractility, but they may also raise the risk of arrhythmias in some patients.
在心脏病学中,PDE3 抑制剂可增强心肌收缩力,但在部分患者中也可能增加心律失常风险。

Etymology / 词源

PDE3 来自科学命名与缩写:PDEphosphodiesterase(磷酸二酯酶)的首字母缩写,后面的 3 表示该酶家族中的第3型/第3类同工酶分组方式。该缩写常用于生物化学、药理学与医学文献中。

Related Words / 相关词

Literary Works / 文学与著作例证

  • Goodman & Gilman’s The Pharmacological Basis of Therapeutics(《古德曼与吉尔曼:药理学原理》)中在强心药与 PDE 抑制剂章节常提及 PDE3
  • Harrison’s Principles of Internal Medicine(《哈里森内科学》)在心力衰竭与相关药物机制部分可见 PDE3
  • Rang & Dale’s Pharmacology(《Rang & Dale 药理学》)在细胞信号与心血管药理内容中会讨论 PDE3 与 cAMP 通路
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