V2EX mln4924

MLN4924

释义 Definition

MLN4924 是一种药物研发代号,后来被命名为 Pevonedistat(佩沃奈司他)。它主要作为NEDD8 激活酶(NAE)抑制剂研究,用于干扰蛋白质的泛素化/降解相关通路,曾在多种癌症(如急性髓系白血病等)的临床研究中出现。该词属于生物医药领域专有名词

发音 Pronunciation (IPA)

/m l n fr nan tu fr/

例句 Examples

MLN4924 is being studied as a potential cancer treatment.
MLN4924 正在被研究作为一种潜在的抗癌治疗药物。

In the trial, MLN4924 inhibited the NEDD8-activating enzyme, disrupting protein regulation pathways and slowing tumor cell growth.
在该试验中,MLN4924 抑制了 NEDD8 激活酶,干扰蛋白调控通路,从而减缓肿瘤细胞生长。

词源 Etymology

MLN4924 属于研发阶段的项目/化合物编号:常见于制药公司或研究机构对候选分子的内部命名体系中。“MLN”通常与早期研发机构/管线标识相关,“4924”为序列编号。该化合物后来以通用名 Pevonedistat 更常见于论文与临床资料。

相关词 Related Words

文学/作品中的用例 Literary Works

由于它是药物研发代号,主要出现于科学论文与临床研究(而非传统文学作品)中,例如:

  • Nature MedicineClinical Cancer ResearchBlood 等期刊中关于 MLN4924/Pevonedistat 的研究论文
  • 与急性髓系白血病(AML)、骨髓增生异常综合征(MDS)等相关的临床研究报道与综述文章
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