V2EX lisdexamfetamine

Lisdexamfetamine

Definition / 释义

利斯的安非他明:一种处方中枢神经兴奋剂,属于前药(prodrug),在体内转化为右旋安非他明(dextroamphetamine)后发挥作用;常用于治疗注意缺陷多动障碍(ADHD),在部分国家/地区也用于中重度暴食症(binge eating disorder)。该词在医学语境中使用更常见。

Pronunciation / 发音

/ls.dk.smft..min/

Examples / 例句

My doctor prescribed lisdexamfetamine for ADHD.
医生给我开了利斯的安非他明来治疗注意缺陷多动障碍。

Because lisdexamfetamine is a prodrug, its effects can feel smoother compared with some immediate-release stimulants.
由于利斯的安非他明属于前药,与一些速释兴奋剂相比,它的作用有时会被描述为更平稳。

Etymology / 词源

该词是一个药物学构词:由 **lisdex-**(可理解为与“赖氨酸 lysine”相关的部分)+ amfetamine(安非他明)组合而成,指这种分子结构把右旋安非他明与氨基酸(赖氨酸)连接,进入体内后再被代谢“释放”出活性成分,因此被称为“前药”。

Related Words / 相关词

Notable Works / 文学与著作中的用例

  • Stahl’s Essential Psychopharmacology(《斯塔尔精神药理学精要》)等精神药理学教材与临床综述中常见该药名,用于讨论ADHD治疗选择与兴奋剂机制。
  • The Maudsley Prescribing Guidelines in Psychiatry(《莫兹利精神科处方指南》)等处方指南类著作中可见,用于剂量、用药监测与注意事项的临床条目。
  • 多篇ADHD与暴食症的随机对照试验与系统综述(医学期刊论文)中频繁出现该术语,作为研究用药与结局指标的一部分。
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