V2EX selinexor

Selinexor

释义 Definition

Selinexor(塞利尼索):一种口服小分子抗肿瘤药物,属于选择性核输出抑制剂(SINE),主要通过抑制核输出蛋白 Exportin 1(XPO1/CRM1),促使某些抑癌蛋白留在细胞核内,从而抑制肿瘤细胞生长。常用于部分血液肿瘤(如多发性骨髓瘤等)的治疗方案中。

发音 Pronunciation

/ slnksr /

例句 Examples

Selinexor is taken by mouth as part of a cancer treatment regimen.
塞利尼索可口服,用作癌症治疗方案的一部分。

In clinical trials, selinexor combined with other agents showed activity in patients with relapsed or refractory multiple myeloma.
在临床试验中,塞利尼索与其他药物联合使用,对复发或难治性多发性骨髓瘤患者显示出一定疗效。

词源 Etymology

Selinexor 是药物的国际非专利名称(INN)。其构词更多是现代药名命名规则下的“可识别且独特”的组合;其中 -exor 常被解读为与其作用靶点相关(与 export/exportin(核输出) 的概念呼应),提示该药与“核输出抑制”机制有关。

相关词 Related Words

文献与作品 Notable Works

  • *Selinexor, Bortezomib, and Dexamethasone for Patients with Multiple Myeloma (BOSTON trial)*(临床研究论文,发表于重要医学期刊)
  • *Selinexor plus low-dose Dexamethasone in Relapsed/Refractory Multiple Myeloma (STORM study)*(关键临床试验相关论文/报道)
  • *U.S. FDA Prescribing Information for XPOVIO (selinexor)*(美国 FDA 药品说明书/审评资料,常被引用的权威医学文本)
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