V2EX active site

Active Site

定义 Definition

Active site(活性位点)是生物化学术语,指酶(enzyme)分子上与底物(substrate)结合并催化化学反应的特定区域。这是酶发挥功能的关键部位。

发音 Pronunciation

/k.tv sat/

例句 Examples

The active site of the enzyme binds to the substrate.
酶的活性位点与底物结合。

A mutation in the active site can dramatically reduce the enzyme's catalytic efficiency, potentially disrupting critical metabolic pathways.
活性位点的突变可能会大幅降低酶的催化效率,从而可能破坏关键的代谢途径。

词源 Etymology

Active 源自拉丁语 activus,意为"有行动力的、积极的",由 agere(做、行动)派生而来。Site 源自拉丁语 situs,意为"位置、场所"。两词组合为生物化学专用术语,最早在20世纪中期随着酶学研究的发展而广泛使用,用来描述酶分子中直接参与催化反应的特定空间区域。

相关词汇 Related Words

文学与学术引用 Literary & Academic References

  • 《Lehninger Principles of Biochemistry》经典生物化学教材,详细阐述了活性位点的结构与功能机制。
  • 《Molecular Biology of the Cell》(Bruce Alberts 等著)在讨论酶催化机制时大量使用该术语。
  • Daniel Koshland 的"诱导契合模型"(Induced Fit Model)论文中,active site 是核心概念,描述酶如何在与底物结合时改变构象以适应反应。
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